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MediCaine MEDICAINE
DERMATOLOGY

PRESCRIPTION NUMBING CREAM FOR DERMATOLOGY

Compounded multi-agent topical anesthetics engineered for dermatologic procedures. Faster onset, deeper penetration, and longer duration than commercial alternatives.

WHY DERMATOLOGISTS CHOOSE COMPOUND ANESTHETICS

Over-the-counter topical anesthetics are limited to a maximum of 4-5% lidocaine. For the procedural demands of a dermatology practice, these concentrations are inadequate. OTC products deliver shallow, short-lived numbness that fails during laser passes, excisions, and deeper tissue work.

Prescription compounded topical anesthetics solve this by combining multiple anesthetic agents at concentrations that far exceed OTC limits. A compounded BLT cream at 20/10/10 delivers three distinct agents through separate pharmacological pathways, producing additive and synergistic anesthesia that a single-agent product cannot match.

Multi-agent formulations also reduce the required concentration of any individual agent, lowering the risk of systemic toxicity while increasing total anesthetic effect at the tissue level. For dermatologists performing back-to-back procedures across large surface areas, this therapeutic index advantage is clinically significant.

HIGHER CONCENTRATIONS

Compounded formulations deliver lidocaine at 10-30%, tetracaine at 7-10%, and benzocaine at 20% -- far beyond OTC ceilings.

MULTI-AGENT SYNERGY

Combining ester and amide anesthetics blocks sodium channels through independent mechanisms for deeper, more reliable numbness.

VASOCONSTRICTION

Phenylephrine 0.5% localizes the anesthetic at the treatment site, extends duration, and reduces procedural bleeding.

CLINICAL APPLICATIONS

DERMATOLOGY PROCEDURES REQUIRING TOPICAL ANESTHESIA

Prescription numbing cream is indicated across the full spectrum of dermatologic procedures. Each procedure type demands specific anesthetic depth, onset timing, and duration.

LASER RESURFACING

Ablative and non-ablative laser resurfacing generates significant thermal discomfort across broad treatment areas. Compound numbing cream applied under occlusion 30-45 minutes prior to the procedure provides consistent anesthesia across the full facial field. Multi-agent formulations maintain efficacy through multiple laser passes.

MOHS SURGERY

While Mohs micrographic surgery relies primarily on injectable local anesthesia, topical compound anesthetic applied prior to the initial injection significantly reduces needle-insertion pain. For patients requiring multiple stages over several hours, reapplication between stages improves comfort during an already lengthy procedure.

SKIN BIOPSIES

Punch biopsies, shave biopsies, and excisional biopsies all benefit from pre-procedural topical anesthesia. Applying prescription lidocaine cream 20-30 minutes before the biopsy reduces or eliminates the need for injectable lidocaine at the biopsy site, streamlining workflow and reducing patient anxiety.

CRYOTHERAPY

Liquid nitrogen cryotherapy for actinic keratoses, warts, and superficial lesions produces sharp, burning discomfort. Pre-treatment with compounded topical anesthetic reduces pain perception during freeze cycles and minimizes the vasovagal response seen in sensitive patients, particularly when treating multiple lesions in a single session.

CHEMICAL PEELS

Medium-depth and deep chemical peels -- including TCA peels and phenol-croton oil formulations -- cause significant stinging and burning during application. Topical anesthesia applied beforehand reduces patient discomfort without interfering with peel penetration, provided the anesthetic is fully removed before acid application.

IPL PHOTOTHERAPY

Intense pulsed light treatments for vascular lesions, pigmentation, and photorejuvenation produce a snapping, heat-based discomfort with each pulse. Pre-treatment topical anesthesia allows higher fluence settings and more aggressive treatment parameters, improving clinical outcomes while maintaining patient comfort throughout the session.

FORMULATIONS

COMPOUND FORMULATIONS EXPLAINED

Understanding the pharmacology behind each compounded formulation and how agent selection affects clinical performance in dermatologic procedures.

BLT

BLT 20/10/10

The most widely prescribed compounded topical anesthetic in dermatology. Benzocaine 20% provides rapid surface-level sodium channel blockade within minutes of application. Lidocaine 10% penetrates deeper tissue layers as an amide anesthetic with a distinct metabolic pathway. Tetracaine 10% extends the duration of numbness with its long half-life. The three agents attack pain signal transmission through complementary mechanisms, producing reliable anesthesia across both superficial and mid-dermal tissue layers. This is the formulation found in MediCaine Pro.

Triple-Agent ~15 Min Onset 2-4 Hr Duration
LT

LT 30/7 HIGH-CONCENTRATION

A dual-agent formulation that maximizes lidocaine concentration at 30% paired with tetracaine at 7%. This approach delivers the deepest tissue penetration of any topical formulation, relying on the high lidocaine load to saturate nerve fibers at depth. The trade-off is a slightly longer onset time compared to BLT and a shorter overall duration window. Ideal for procedures requiring maximum depth of anesthesia over a focused area. This is the formulation found in MediCaine Elite.

Dual-Agent ~20 Min Onset 1-3 Hr Duration
BLT+

QUAD-AGENT BLT+ WITH PRILOCAINE

The maximum-potency formulation adds prilocaine 8% as a fourth anesthetic agent to the BLT base. Prilocaine is an amide anesthetic that works synergistically with lidocaine while blocking sodium channels at a different binding site. The result is the most comprehensive topical anesthesia available without injection -- four independent agents creating overlapping numbness across all tissue depths with the longest duration window. Phenylephrine 0.5% is included as a vasoconstrictor to localize the agents and reduce procedural bleeding. This is the formulation found in MediCaine Ultra.

Quad-Agent ~15 Min Onset 3-5 Hr Duration
COMPARISON

COMPOUNDED VS COMMERCIAL PRODUCTS

How MediCaine compounded formulations compare to EMLA, Pliaglis, and other commercially available topical anesthetics used in dermatology.

MEDICAINE COMPOUND

Compounded BLT / LT / BLT+

Up to 4 anesthetic agents at prescription-strength concentrations
15-minute onset with BLT formulations
Up to 5 hours of anesthetic duration
Vasoconstrictor included (Pro and Ultra)
Compounded fresh per order, not mass-manufactured
Airless pump packaging for precise, hygienic dosing
EMLA

Lidocaine 2.5% / Prilocaine 2.5%

Only 5% total anesthetic concentration
60-minute onset required for adequate anesthesia
1-2 hour duration at best
No vasoconstrictor -- causes vasodilation
Shallow penetration, insufficient for laser procedures
Methemoglobinemia risk with large-area application
PLIAGLIS

Lidocaine 7% / Tetracaine 7%

14% total concentration -- better than EMLA but below compounded BLT
20-30 minute onset with peel-off delivery system
Only 2 anesthetic agents, no benzocaine surface blockade
No vasoconstrictor
Significantly higher cost per application
Fixed formulation -- cannot be customized for specific procedures
FAQ

NUMBING CREAM FOR DERMATOLOGY

What numbing cream do dermatologists use for procedures?+
Dermatologists use compounded prescription topical anesthetics for procedural pain management. The most common formulations are BLT (Benzocaine 20%, Lidocaine 10%, Tetracaine 10%) and LT (Lidocaine 30%, Tetracaine 7%). These multi-agent compounds deliver significantly higher anesthetic concentrations than over-the-counter products, with onset in 15-20 minutes and duration of 2-5 hours depending on the formulation. MediCaine offers three tiers -- Pro (BLT), Elite (LT), and Ultra (BLT+ with Prilocaine) -- to match the anesthetic demands of different dermatologic procedures.
Is compounded lidocaine tetracaine cream better than EMLA?+
Yes. EMLA contains only Lidocaine 2.5% and Prilocaine 2.5% -- a total of 5% anesthetic concentration -- and requires 60 minutes of application for adequate anesthesia with a duration of 1-2 hours. Compounded lidocaine tetracaine cream delivers substantially higher concentrations: MediCaine Elite provides Lidocaine 30% and Tetracaine 7% (37% total), while MediCaine Pro delivers Benzocaine 20%, Lidocaine 10%, and Tetracaine 10% (40% total). The compounded formulations achieve onset in 15-20 minutes, penetrate deeper tissue layers, and maintain anesthesia for 2-5 hours. EMLA also causes vasodilation at the treatment site, whereas MediCaine Pro and Ultra include Phenylephrine as a vasoconstrictor to reduce procedural bleeding.
How long should numbing cream be applied before a laser procedure?+
For laser procedures, apply compound numbing cream 20-30 minutes before treatment under occlusive dressing (plastic wrap or Tegaderm). The occlusion enhances percutaneous absorption and drives the anesthetic agents deeper into the dermal tissue. For ablative laser resurfacing and deep fractional treatments, a full 30-minute application under occlusion is recommended. For non-ablative laser and IPL, 20 minutes is typically sufficient. Remove the numbing cream completely and clean the treatment area before beginning laser passes.
Do I need a prescription for compound numbing cream?+
MediCaine compound numbing cream is available exclusively to licensed healthcare providers. Orders require NPI (National Provider Identifier) verification, which is completed electronically during the ordering process using the NPI Registry. This verification confirms your active medical license and authorizes the compounding pharmacy to prepare prescription-strength formulations for your practice. Licensed dermatologists, physician assistants, nurse practitioners, and other qualified providers can order directly through the online configurator or by calling (310) 889-0733.
What is the strongest numbing cream for dermatology?+
MediCaine Ultra is the strongest topical anesthetic available for dermatologic procedures. It is a quad-agent formulation containing Benzocaine 20%, Lidocaine 10%, Tetracaine 10%, and Prilocaine 8%, with Phenylephrine 0.5% as a vasoconstrictor. The four independent anesthetic agents block sodium channels through separate pharmacological pathways, producing the most comprehensive topical anesthesia available without injection. Ultra provides onset in approximately 15 minutes and duration of 3-5 hours. It is recommended for ablative laser resurfacing, deep chemical peels, and extended multi-stage dermatologic procedures.

ORDER FOR YOUR PRACTICE

Compounded fresh per order in the USA. Available in cream or ointment, with airless pump or jar packaging.

Licensed providers can order directly through our configurator or call our pharmacist to discuss formulation recommendations for your procedure mix.